2021

Krajcovicova, S.; Hlavac, J.; Vychodilova, K.
Polymer-supported synthesis of N-substituted anthranilates as the building blocks for preparation of N-arylated 3-hydroxyquinolin-4(1H)-ones
RSC Adv., 2021, 11, 9362-9365.

Vanda, D.; Canale, V.; Chaumont-Dubel, S.; Kurczab, R.; Satała, G.; Koczurkiewicz, P.; Krawczyk, M.; Pietruś, W.; Blicharz, K.; Pękala, E.; Bojarski, A.; Popik, P.; Marin, P.; Soural, M.; Zajdel, P.
Imidazopyridine-based 5-HT6 receptor neutral antagonists: impact of N1-benzyl and N1-phenylsulfonyl fragments on different receptor conformational state
J. Med. Chem. 202164, 1180-1196.

Kriegelsteinova, P.; Lemrova, B.; Rucilova, V.; Soural, M.
Copper-free solid-phase synthesis of triazolo[1,5-a][1,4]diazepin-6-ones
Adv. Synth. Catal. 2021363, 1112-1119.

Krajcovicova, S.; Jorda, R.; Vanda, D.; Soural, M.; Krystof, V.
1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton’s tyrosine kinase
Eur. J. Med. Chem., 2021, 211, 113094.

Rucilova, V.; Swierczek, A.; Vanda, D.; Funk, P.; Lemrova, B.; Gawalska, A.; Bucki, A.; Nowak, B.; Zadrozna, M.; Pociecha, K.; Soural, M.; Wyska, E.; Pawlowski, M.; Chlon-Rzepa, G.; Zajdel, P.
New Imidazopyridines with Phosphodiesterase 4 and 7 Inhibitory Activity and Their Efficacy in Animal Models of Inflammatory and Autoimmune Diseases
Eur. J. Med. Chem., 2021, 209, 112854.